{"id":142802,"date":"2025-05-12T13:48:37","date_gmt":"2025-05-12T13:48:37","guid":{"rendered":"https:\/\/www.unipi.it\/ateneo\/organizzazione\/persone\/simone-brogi-136018-en\/"},"modified":"2026-04-01T04:34:02","modified_gmt":"2026-04-01T02:34:02","slug":"simone-brogi-136018-en","status":"publish","type":"unipi_persone","link":"https:\/\/www.unipi.it\/en\/about-us\/organisation\/people\/simone-brogi-136018-en\/","title":{"rendered":"Simone Brogi"},"content":{"rendered":"<p>Professore Associato &#8211; Dipartimento di Farmacia | Tel.: 050 2219613 &#8211; Email: simone.brogi@unipi.it<\/p>\n","protected":false},"template":"","meta":{"unipi-persone-chiave":"136018","unipi-persone-nome":"Simone","unipi-persone-cognome":"Brogi","unipi-persone-email":"simone.brogi@unipi.it","unipi-persone-cv":"","unipi-persone-link-esterno-cv":"https:\/\/www.researchgate.net\/profile\/Simone_Brogi","unipi-persone-modalita-ricevimento":"","unipi-persone-luogo-ricevimento":"","unipi-persone-ore-ricevimento":"","unipi-persone-telefono":"050 2219613","unipi-persone-sitoweb":"","unipi-persone-cariche":"","unipi-persone-link-orario-lezioni":"https:\/\/unipi.prod.up.cineca.it\/calendarioPubblico\/matricola=041495","unipi-persone-link-registro-lezioni":"https:\/\/unimap.unipi.it\/registri\/registri.php?ri=041495&tmplt=principale.tpl","unipi-persone-settore-scientifico":"Farmacologia BIOS-11\/A","unipi-persone-ruolo":"Professore Associato","unipi-persone-arpi":"https:\/\/arpi.unipi.it\/cris\/rp\/rp99264","unipi-persone-pubblicazioni":"<ul class=\"pubblicazioni-list\"><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1355027\" target=\"_blank\" rel=\"noopener noreferrer\">Discovery of thieno[2,3-d]pyrimidine-based dual Aurora B\/VEGFR-2 inhibitors with potent anticancer activity: molecular docking, mechanistic studies, and in vivo validation in a breast cancer model<\/a> <span class=\"pub-details\">(El-Shafey, H. W.; Hamdi, A.; Elnagar, M. R.; Gebril, S. M.; Haikal, A.; El-Azab, A. S.; Brogi, S.; Al-Suwaidan, I. A.; Abdel-Aziz, A. A. -M. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1354487\" target=\"_blank\" rel=\"noopener noreferrer\">Quinazoline-sulfonamide hybrids as multitarget anticancer agents: inhibition of carbonic anhydrase IX\/XII isoforms and VEGFR-2 with in vitro and in silico validation<\/a> <span class=\"pub-details\">(Zeidan, M. A.; Al-Sanea, M. M.; Elnagar, M. R.; Tawfik, M. M.; El-Shafey, H. W.; Tawfik, S. S.; Brogi, S.; Hamdi, A. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1353567\" target=\"_blank\" rel=\"noopener noreferrer\">2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition<\/a> <span class=\"pub-details\">(Cernicchi, G.; Nizi, M. G.; Emmolo, R.; Persoons, L.; Laporte, M.; Jochmans, D.; Romeo, I.; Pepe, G.; Milite, C.; Campiglia, P.; Spezzini, J.; Martelli, A.; Brogi, S.; Esposito, F.; Felicetti, T.; Massari, S.; Manfroni, G.; Sabatini, S.; Sbardella, G.; Alcaro, S.; Neyts, J.; Corona, A.; Tramontano, E.; De Jonghe, S.; Tabarrini, O. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1352627\" target=\"_blank\" rel=\"noopener noreferrer\">Dimeric Anthraquinone Rugulosin A Induces Apoptosis in Lung Adenocarcinoma and Targets PI3K\/AKT\/MAPK Pathways In Silico<\/a> <span class=\"pub-details\">(Manzano, J. A. H.; Abellanosa, E. A. M.; Aguilar, J. P. P.; Brogi, S.; Yen, C. -H.; Notarte, K. I.; Austriaco, N.; Macabeo, A. P. G. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1351847\" target=\"_blank\" rel=\"noopener noreferrer\">Second-generation prokineticin PKR1 receptor agonists: Advancing cardioprotection against chemotherapy-induced toxicity<\/a> <span class=\"pub-details\">(Audebrand, A.; Brogi, S.; Tezeren, M.; Tafi, A.; Ocak, O. H.; Koyuncu, H.; Tetko, I.; Desaubry, L.; Nebigil, C. G. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1350448\" target=\"_blank\" rel=\"noopener noreferrer\">Quinazolinone-Based PqsR Modulators Suppress Quorum-Sensing\u2013Driven Virulence in Pseudomonas aeruginosa<\/a> <span class=\"pub-details\">(Tudino, V.; Mellini, M.; Milioni, L.; Carullo, G.; Rossi, S.; Giammarino, F. M. P. R.; Butini, S.; Brogi, S.; Ciccone, V.; Visca, P.; Leoni, L.; Rampioni, G.; Gemma, S.; Campiani, G. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1345847\" target=\"_blank\" rel=\"noopener noreferrer\">Targeting Class I Histone Deacetylases Triggers Antitumor Responses in Colorectal Cancer In Vitro and In Vivo<\/a> <span class=\"pub-details\">(Carullo, G.; Falbo, F.; Tudino, V.; Song, J.; Fava, M.; Fontana, A.; Koch, A.; Heiss, A.; Erlenbach-Wuensch, K.; Panzeca, G.; Brogi, S.; Bichicchi, A.; Saponara, S.; Fusi, F.; Vincenzi, F.; Varani, K.; Cappello, M.; Pasquini, S.; Ramunno, A.; Pepe, G.; Butini, S.; Aiello, F.; Gemma, S.; Schneider-Stock, R.; Campiani, G. - 2026 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1337473\" target=\"_blank\" rel=\"noopener noreferrer\">In Silico Exploration of Potential Inhibitors Targeting SARS-CoV-2 Non-Structural Protein 15 [Nsp15]: A Comprehensive Overview of Current Research<\/a> <span class=\"pub-details\">(Yazdani, B.; Sirous, H.; Farzam, F.; Ansarizadeh, S.; Karimi Taheri, M.; Pourmohammad-Hosseini, G.; Noei, M.; Daneshipour, K.; Shakeri, D.; Houshangi, M.; Calderone, V.; Brogi, S. - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1334947\" target=\"_blank\" rel=\"noopener noreferrer\">Exploiting COX-2 engagement for amplifying anticancer potential of Quinazoline-triazole conjugates with superior EGFR\/VEGFR-2 inhibition<\/a> <span class=\"pub-details\">(Serag, M. I.; Hamdi, A.; Nasr, E. E.; Elnagar, M. R.; Tawfik, M. M.; El-Azab, A. S.; Brogi, S.; Al-Suwaidan, I. A.; Hefnawy, M.; Abdel-Aziz, A. A. -M. - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1334268\" target=\"_blank\" rel=\"noopener noreferrer\">Pharmacological Investigation of a Novel Resveratrol-like SIRT1 Activator Endowed with a Cardioprotective Profile<\/a> <span class=\"pub-details\">(Carbonetti, Leonardo; Brogi, Simone; D&#039;Orsi, Rosarita; Lessi, Marco; Calderone, Vincenzo; Testai, Lara; Bellina, Fabio - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1323487\" target=\"_blank\" rel=\"noopener noreferrer\">Uncovering a Mutation-Independent Therapeutic Strategy against Inherited Retinal Diseases: Development of Class I HDAC\/LSD1 Hybrid Inhibitors<\/a> <span class=\"pub-details\">(Carullo, G.; Piano, I.; Salamone, G.; Corsi, F.; Orsini, N.; Dichiara, M.; Cursaro, I.; Fontana, A.; Galante, A.; Contri, C.; Guadagno, L.; Caroli, J.; Mattevi, A.; Vincenzi, F.; Varani, K.; Brogi, S.; Gemma, S.; Butini, S.; Gargini, C.; Strettoi, E.; Campiani, G. - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1322729\" target=\"_blank\" rel=\"noopener noreferrer\">Hydroxyl carboxylic acid receptor-2 [HCAR2] as a potential target in neurometabolic diseases<\/a> <span class=\"pub-details\">(Testai, Lara; Guida, Francesca; Salerno, Silvia; Brogi, Simone; Morace, Andrea Maria; Carbonetti, Leonardo; Ricciardi, Federica; Perrone, Michela; Palazzo, Enza; Calderone, Vincenzo; Maione, Sabatino; Luongo, Livio - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1322657\" target=\"_blank\" rel=\"noopener noreferrer\">DNA gyrase-inhibitory antimicrobial anthraquinone from the endophytic Sordariomycetes fungus Diaporthe perseae<\/a> <span class=\"pub-details\">(Manzano, Joe Anthony H.; Abanto, John Cyril D.; Dayo, Beaver Andrei F.; Llames, Lloyd Christian J.; Gonzaga, Mary Grace E.; Brogi, Simone; Macabeo, Allan Patrick G. - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1317030\" target=\"_blank\" rel=\"noopener noreferrer\">Editorial: Pharmacokinetics modeling in the Artificial Intelligence Era<\/a> <span class=\"pub-details\">(Brogi, S.; Schyman, P.; Siramshetty, V. B. - 2025 - 1.1 Articolo in rivista)<\/span><\/li><li><a href=\"https:\/\/arpi.unipi.it\/handle\/11568\/1313647\" target=\"_blank\" rel=\"noopener noreferrer\">Novel Antiviral Agents: Synthesis, Molecular Modelling Studies and Biological Investigation, 2nd Edition<\/a> <span class=\"pub-details\">(Brogi, S. - 2025 - 1.1 Articolo in rivista)<\/span><\/li><\/ul>","unipi-persone-didattica":"<ul class=\"registri-list\"><li>Modulo ii (modulo dell'insegnamento il principio delle 3r negli studi preclinici: dai tessuti ricostituiti agli approcci computazionali cod. 007ce) per Laurea Magistrale Ciclo Unico 5 anni in Chimica e tecnologia farmaceutiche<br\/><strong>Insegnamenti condivisi\/mutuati:<\/strong><ul class=\"registri-shared\"><li>Il principio delle 3r negli studi preclinici: dai tessuti ricostituiti agli approcci computazionali (cod. 007CE) - Laurea Magistrale Ciclo Unico 5 anni in Chimica e tecnologia farmaceutiche<\/li><\/ul><\/li><li>Farmacognosia (modulo dell'insegnamento farmacologia e farmacognosia cod. 398ee) per Laurea in Scienze dei prodotti erboristici e della salute<\/li><li>Farmaci e integratori alimentari in ambito sportivo (cod. 0007E) per Laurea Magistrale in Scienze della nutrizione umana<\/li><\/ul>","unipi-persone-codocenze":"<h4 class=\"mt-2\">Incarichi di co-docenza in moduli\/insegnamenti<\/h4><ul><li>Nutraceutica e Nutrigenomica (Cod. 003EG) per Laurea Magistrale in Scienze della nutrizione umana<\/li><li>Farmacognosia e Tossicologia (Modulo dell&#039;insegnamento Farmacologia, Farmacoterapia, Farmacognosia e Tossicologia Cod. 464EE) per Laurea Magistrale Ciclo Unico 5 anni in Chimica e tecnologia farmaceutiche<\/li><\/ul>","unipi-persone-interessi-ricerca":"","_wpml_word_count":"13","_last_translation_edit_mode":"translation-editor","unipi-persone-dati-posizione":"","_elementor_page_assets":[]},"organizzazioni":[3628],"class_list":["post-142802","unipi_persone","type-unipi_persone","status-publish","hentry","organizzazioni-dipartimento-di-farmacia-449999-en"],"email":"simone.brogi@unipi.it","telefono":"050 2219613","content_plain":"Professore Associato &#8211; 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